Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Epidermal growth factor receptor' and Ligand = 'BDBM149409'
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Celgene Avilomics Research, Inc.

US Patent
LigandPNGBDBM149409(US10434101, Compound I-9 | US11096942, Compound I-...)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.5Assay Description:Briefly, 10x stocks of EGFR-WT (PV3872) from Invitrogen and EGFR-T790M/L858R (40350) from BPS Bioscience, San Diego, Calif., 1.13xATP (AS001A) and ap...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2DVSUS Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Celgene Avilomics Research, Inc.

US Patent
LigandPNGBDBM149409(US10434101, Compound I-9 | US11096942, Compound I-...)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Briefly, 10× stocks of EGFR-WT (PV3872) from Invitrogen and EGFR-T790M/L858R (40350) from BPS Bioscience, San Diego, Calif., 1.13×ATP (AS001A) and ap...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GT5RBQUS Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Celgene Avilomics Research, Inc.

US Patent
LigandPNGBDBM149409(US10434101, Compound I-9 | US11096942, Compound I-...)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Briefly, 10× stocks of EGFR-WT (PV3872) from Invitrogen and EGFR-T790M/L858R (40350) from BPS Bioscience, San Diego, Calif., 1.13×ATP (AS001A) and ap...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3HD3US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Celgene Avilomics Research, Inc.

US Patent
LigandPNGBDBM149409(US10434101, Compound I-9 | US11096942, Compound I-...)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMpH: 7.5Assay Description:Briefly, 10x stocks of EGFR-WT (PV3872) from Invitrogen and EGFR-T790M/L858R (40350) from BPS Bioscience, San Diego, Calif., 1.13xATP (AS001A) and ap...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2DVSUS Patent