Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM263664'
TargetEstrogen receptor(Homo sapiens (Human))
SANOFI

US Patent
LigandPNGBDBM263664(US9714221, Example 1)copy SMILEScopy InChI
Affinity DataIC50: 7nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N58PB1US Patent
TargetEstrogen receptor(Homo sapiens (Human))
SANOFI

US Patent
LigandPNGBDBM263664(US9714221, Example 1)copy SMILEScopy InChI
Affinity DataEC50:  0.400nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed