Found 5 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM263669' TargetEstrogen receptor(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Ability to inhibit the rat muscle adenylate kinase lII in competition with the AMP variedMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Beta-2 adrenergic receptor antagonistic activity on guinea pig tracheal chainsMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Antagonist activity at recombinant human His6-tagged ERalpha LBD (298 to 554 residues) Y537S mutant expressed in Escherichia coli assessed as inhibit...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity at recombinant human His6-tagged ERalpha LBD (298 to 554 residues) D538G mutant expressed in Escherichia coli assessed as inhibit...More data for this Ligand-Target Pair
