Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM263913'
TargetEstrogen receptor(Homo sapiens (Human))
SANOFI

US Patent
LigandPNGBDBM263913(6-(4- chloro- phenyl)-5-[4- [(3S)-1-(3- fluoroprop...)copy SMILEScopy InChI
Affinity DataIC50: 11nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N58PB1US Patent
TargetEstrogen receptor(Homo sapiens (Human))
SANOFI

US Patent
LigandPNGBDBM263913(6-(4- chloro- phenyl)-5-[4- [(3S)-1-(3- fluoroprop...)copy SMILEScopy InChI
Affinity DataEC50:  8nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed