Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM50090463'
TargetEstrogen receptor(Homo sapiens (Human))
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50090463(CHEMBL3581633)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Displacement of fluormone-labeled ES2 from recombinant full length human ERalpha ligand binding domain expressed in insect cells after 2 hrs by TR-FR...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J10557PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50090463(CHEMBL3581633)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Downregulation of ERalpha in human MCF7 cells after 4 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J10557PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50090463(CHEMBL3581633)copy SMILEScopy InChI
Affinity DataEC50:  113nMAssay Description:Induction of estrogen receptor-alpha degradation in human MCF7 cells after 4 hrs by in-cell western assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0H7QPubMed