Affinity DataIC50: 14nMAssay Description:Displacement of fluormone-labeled ES2 from recombinant full length human ERalpha ligand binding domain expressed in insect cells after 2 hrs by TR-FR...More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Downregulation of ERalpha in human MCF7 cells after 4 hrs by Western blot analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 113nMAssay Description:Induction of estrogen receptor-alpha degradation in human MCF7 cells after 4 hrs by in-cell western assayMore data for this Ligand-Target Pair