Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM50234790'
TargetEstrogen receptor(Homo sapiens (Human))
Universita di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)copy SMILEScopy InChI
Affinity DataKi:  310nMAssay Description:Displacement of [3H]estradiol from purified full length human ERalpha receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ40SBPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Universita di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)copy SMILEScopy InChI
Affinity DataEC50:  26nMAssay Description:Agonist activity at full length human ERalpha receptor expressed in human HEC-1 cells assessed as (ERE)2-pS2-luc reporter gene transcriptional activi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ40SBPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Universita di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)copy SMILEScopy InChI
Affinity DataEC50:  26nMAssay Description:Agonist activity at full-length human estrogen receptor alpha expressed in human HEC1 cells assessed as transcriptional activation after 24 hrs by lu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0SRHPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Universita di Pisa

Curated by ChEMBL
LigandPNGBDBM50234790((E)-2-chloro-3,4'-dihydroxybiphenyl-4-carbaldehyde...)copy SMILEScopy InChI
Affinity DataEC50:  26nMAssay Description:Agonist activity at full-length human estrogen receptor alpha expressed in human HEC1 cells assessed as transcriptional activation after 24 hrs by lu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0SRHPubMed