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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Estrogen receptor [Y537S]' and Ligand = 'BDBM263737'
Target
Estrogen receptor [Y537S]
(Homo sapiens (Human))
SANOFI
US Patent
Ligand
BDBM263737
(6-(6- ethoxy-2- fluoro-3- pyridyl)-5- [4-[(3S)- 1-...)
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Affinity Data
IC50: 18nM
pH: 7.4 T: 2°C
Assay Description:
It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2N58PB1
US Patent