Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Extracellular calcium-sensing receptor' and Ligand = 'BDBM50261666'
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Enteroendocrine Discovery Performance Unit and Platform Technologies and Science, GlaxoSmithKline, 5 Moore Drive, Research Triangle Park, NC 27709, United States. Electronic address: ssparks@viamet.c

Curated by ChEMBL
LigandPNGBDBM50261666(CHEMBL4100132)copy SMILEScopy InChI
Affinity DataEC50:  16nMAssay Description:Agonist activity at human beta-2 adrenergic receptor expressed in human H292 cells assessed as accumulation of intracellular cAMP after 1 hr by Alpha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889FRPubMed