Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Fibroblast growth factor receptor 3' and Ligand = 'BDBM261919'
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Incyte Corporation

US Patent
LigandPNGBDBM261919(2′-(2,6-difluoro-3,5-dimethoxyphenyl)-6̸...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:FGFR1, FGFR2, and FGFR4 are measured under equivalent conditions with the following changes in enzyme and ATP concentrations: FGFR1, 0.02 nM and 210 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TX3HD3US Patent
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Incyte Corporation

US Patent
LigandPNGBDBM261919(2′-(2,6-difluoro-3,5-dimethoxyphenyl)-6̸...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24M97QSUS Patent
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Incyte Corporation

US Patent
LigandPNGBDBM261919(2′-(2,6-difluoro-3,5-dimethoxyphenyl)-6̸...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2G73HS1US Patent
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Incyte Corporation

US Patent
LigandPNGBDBM261919(2′-(2,6-difluoro-3,5-dimethoxyphenyl)-6̸...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC9298US Patent