Compile Data Set for Download or QSAR
Found 7 Enz. Inhib. hit(s) with Target = 'Fibroblast growth factor receptor 4' and Ligand = 'BDBM50525939'
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50525939(Balversa | Erdafitinib | Jnj-42756493)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8WX6PubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50525939(Balversa | Erdafitinib | Jnj-42756493)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Inhibition of recombinant non-phosphorylated FGFR4 kinase domain (442 to 753) (unknown origin) expressed in Sf9 insect cells using 5-Fluo-Ahx-KKKKEEI...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB56MJPubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50525939(Balversa | Erdafitinib | Jnj-42756493)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Inhibition of human FGFR4 incubated for 45 mins by time-resolved fluorescence kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GHPPubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50525939(Balversa | Erdafitinib | Jnj-42756493)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Inhibition of FGFR4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6PWNPubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50525939(Balversa | Erdafitinib | Jnj-42756493)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44HQPubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50525939(Balversa | Erdafitinib | Jnj-42756493)copy SMILEScopy InChI
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49VVSPubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50525939(Balversa | Erdafitinib | Jnj-42756493)copy SMILEScopy InChI
Affinity DataIC50: 19nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765KCQPubMed