Affinity DataEC50: 33nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by aequorin assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.60nMAssay Description:Agonist activity at human GPR40 expressed in mouse A9 cells by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 29nMAssay Description:Agonist activity at cynomolgus monkey GPR40 in presence of 0.01% human serum albumin relative to AMG 837More data for this Ligand-Target Pair
Affinity DataEC50: 33nMAssay Description:Partial agonist activity at human GPR40 expressed in CHO cells measured over 20 secs interval by luminometric analysis in presence of 0.01% human ser...More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:Partial agonist activity at human GPR40 expressed in CHO cells measured over 20 secs interval by luminometric analysis in presence of 100% human seru...More data for this Ligand-Target Pair