Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Furin' and Ligand = 'BDBM50448478'
TargetFurin(Homo sapiens (Human))TBA
LigandPNGBDBM50448478(CHEMBL3126396)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Inhibition of recombinant soluble human furin using pyroGlu-Arg-Thr-Lys-Arg-methyl-coumaryl-7-amide as substrate measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN77KRPubMed
TargetFurin(Homo sapiens (Human))TBA
LigandPNGBDBM50448478(CHEMBL3126396)copy SMILEScopy InChI
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26H4NG9PubMed
TargetFurin(Homo sapiens (Human))TBA
LigandPNGBDBM50448478(CHEMBL3126396)copy SMILEScopy InChI
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26H4NG9PubMed
TargetFurin(Homo sapiens (Human))TBA
LigandPNGBDBM50448478(CHEMBL3126396)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Competitive inhibition of recombinant furin (unknown origin) using as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M09FJPubMed