Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'G protein-coupled receptor kinase 5' and Ligand = 'BDBM50529469'
TargetG protein-coupled receptor kinase 5(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50529469(CHEMBL4456539)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of human GRK5 using tubulin as substrate measured after 30 mins by [gamma-32P]-ATP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3HR8PubMed
TargetG protein-coupled receptor kinase 5(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50529469(CHEMBL4456539)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of human GRK5 using tubulin as substrate measured after 60 mins by [gamma-32P]-ATP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3HR8PubMed
TargetG protein-coupled receptor kinase 5(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50529469(CHEMBL4456539)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Inhibition of human GRK5 using tubulin as substrate measured after 0 mins by [gamma-32P]-ATP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3HR8PubMed