Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'G protein-coupled receptor kinase 5' and Ligand = 'BDBM50566199'
TargetG protein-coupled receptor kinase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50566199(CHEMBL4791260)copy SMILES
Affinity DataKi:  1.00E+3nMAssay Description:Covalent inhibition of GRK5 (unknown origin) using porcine brain tubulin as substrate by [gamma32P]ATP based radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75M3VPubMed
TargetG protein-coupled receptor kinase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50566199(CHEMBL4791260)copy SMILES
Affinity DataIC50: 220nMAssay Description:Inhibition of human GRK5 using porcine brain tubulin as substrate incubated for 3 to 5 mins by [gamma32P]ATP based radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75M3VPubMed