BindingDB PrimarySearch

Found 1 Enz. Inhib. hit(s) with Target = 'Gamma-aminobutyric acid (GABA) B receptor 1/type B receptor subunit 2 [41-940]' and Ligand = 'BDBM24195'

Gamma-aminobutyric acid (GABA) B receptor 1/type B receptor subunit 2 [41-940](Rattus norvegicus (rat))
AstraZeneca

BDBM24195(3-aminopropylphosphinic derivative, (R)-7 | AZD335...)copy SMILEScopy InChI

Ki: 5.10nM ΔG°: -46.9kJ/mole EC50: 8.64nMpH: 7.4 T: 2°CAssay Description:Inhibition of [3H]GABA binding at GABAB receptor sites in rat brain synaptic membranes by test compounds was measured using a filtration binding assa...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article
BindingDB Entry DOI: 10.7270/Q2M32T2TPubMed