Found 5 Enz. Inhib. hit(s) with Target = 'Gamma-aminobutyric acid receptor subunit alpha-5' and Ligand = 'BDBM50049736' TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Moltech Corporation
Curated by ChEMBL
Moltech Corporation
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Binding affinity to GABAA alpha-5-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5(RAT)
University of Wisconsin-Milwaukee
Curated by ChEMBL
University of Wisconsin-Milwaukee
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of [3H]flunitrazepam binding to high affinity GABA-A receptor of rat hippocampal membranesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5(RAT)
University of Wisconsin-Milwaukee
Curated by ChEMBL
University of Wisconsin-Milwaukee
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of [3H]-flunitrazepam binding to alpha5 GABA-A receptor of rat hippocampal membranesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5(RAT)
University of Wisconsin-Milwaukee
Curated by ChEMBL
University of Wisconsin-Milwaukee
Curated by ChEMBL
Affinity DataIC50: 67.2nMAssay Description:Inhibition of [3H]-flunitrazepam binding to alpha5 GABA-A receptor of rat hippocampal membranesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Moltech Corporation
Curated by ChEMBL
Moltech Corporation
Curated by ChEMBL
Affinity DataEC50: 9.80E+3nMAssay Description:Activity at alpha-5-beta-3-gamma-2 GABAA receptor expressed in Xenopus oocytes assessed as inhibition in GABA-induced current by voltage clamp assayMore data for this Ligand-Target Pair
