Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Gamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2' and Ligand = 'BDBM50157997'
LigandPNGBDBM50157997(Butane-1-sulfonic acid tricyclo[8.2.1.0*3,8*]tride...)copy SMILEScopy InChI
Affinity DataIC50: 610nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445KZQPubMed