Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Gastrin/cholecystokinin type B receptor' and Ligand = 'BDBM50008170'
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Merck Sharp& Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008170(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of binding of [125I]gastrin to Cholecystokinin type B receptor from guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29K4BTPPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Rotta Research Laboratorium

Curated by ChEMBL
LigandPNGBDBM50008170(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XS5W11PubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Merck Sharp& Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008170(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+4nMAssay Description:Concentration required to inhibit by 50% the specific binding of [3H]pentagastrin to cholecystokinin type B receptor in rabbit gastric glandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XS5W11PubMed