Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Ligand = 'BDBM50326936'
TargetGlucocorticoid receptor(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals Inc.

Curated by ChEMBL
LigandPNGBDBM50326936(1,1,1-Trifluoro-4-(5-fluoro-2-methoxyphenyl)-4-met...)copy SMILEScopy InChI
Affinity DataIC50: 7.30nMAssay Description:Binding affinity to glucocorticoid receptor expressed in baculovirus-infected insect cells using tetramethylrhodamine labeled Dexamethasone by fluore...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571D0XPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals Inc.

Curated by ChEMBL
LigandPNGBDBM50326936(1,1,1-Trifluoro-4-(5-fluoro-2-methoxyphenyl)-4-met...)copy SMILEScopy InChI
Affinity DataIC50: 8.20nMAssay Description:Transrepression activity at glucocorticoid receptor in HFF assessed as inhibition of IL-1-induced IL-6 production after 18 to 24 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571D0XPubMed