Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Glucokinase regulatory protein' and Ligand = 'BDBM50009118'
TargetGlucokinase regulatory protein(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50009118(CHEMBL3238313)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of biotin-tagged human GKRP/fluorescein-tagged GK interaction preincubated for 20 mins prior to GK addition measured after 2 to 4 hrs by A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V126BFPubMed
TargetGlucokinase regulatory protein(Mus musculus)
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50009118(CHEMBL3238313)copy SMILEScopy InChI
Affinity DataEC50:  349nMAssay Description:Inhibition of GKRP-GK interaction in mouse hepatocytes assessed as induction of GK translocation from nucleus to cytoplasm incubated for 20 mins prio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V126BFPubMed