Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Glutamate carboxypeptidase 2' and Ligand = 'BDBM456906'
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
THE JOHNS HOPKINS UNIVERSITY

US Patent
LigandPNGBDBM456906(US10736974, Compound XY-26 | US10736974, Entry 9)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29C71GJUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
THE JOHNS HOPKINS UNIVERSITY

US Patent
LigandPNGBDBM456906(US10736974, Compound XY-26 | US10736974, Entry 9)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29C71GJUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
THE JOHNS HOPKINS UNIVERSITY

US Patent
LigandPNGBDBM456906(US10736974, Compound XY-26 | US10736974, Entry 9)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29C71GJUS Patent