Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, NMDA 1/2A' and Ligand = 'BDBM10487'
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))TBA
LigandPNGBDBM10487(1-chloro-6H,7H,8H,9H,10H-cyclohepta[b]quinolin-11-...)copy SMILEScopy InChI
Affinity DataIC50: 7.29E+3nMAssay Description:Inhibition of human GluN1a/GluN2A receptor expressed in HEK293 cells assessed as inhibition of glycine/glutamate-induced current measured at -60 mV h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC365GPubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))TBA
LigandPNGBDBM10487(1-chloro-6H,7H,8H,9H,10H-cyclohepta[b]quinolin-11-...)copy SMILEScopy InChI
Affinity DataIC50: 1.12E+5nMAssay Description:Inhibition of human GluN1a/GluN2A receptor expressed in HEK293 cells assessed as relative inhibition of glycine/glutamate-induced current measured at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC365GPubMed