Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, kainate 1' and Ligand = 'BDBM50399431'
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50399431(CHEMBL2178919)copy SMILEScopy InChI
Affinity DataIC50: 0.280nMAssay Description:Antagonist activity at rat GluK1 receptor expressed in Xenopus oocytes by two-electrode voltage-clamp at membrane potential -60 to -80 mV electrophys...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7PXRPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50399431(CHEMBL2178919)copy SMILEScopy InChI
Affinity DataIC50: 0.820nMAssay Description:Antagonist activity at rat GluK1 receptor expressed in Xenopus oocytes at membrane potential -60 mV by two-electrode voltage-clamp electrophysiology ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7PXRPubMed