Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, kainate 3' and Ligand = 'BDBM17657'
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)copy SMILEScopy InChI
Affinity DataKi:  490nMAssay Description:Displacement of [3H]SYM2081 from rat iGluR7 receptor expressed in Sf9 cells baculovirus system after 1 to 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR206GPubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)copy SMILEScopy InChI
Affinity DataKi:  494nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR7More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8DP6PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Universit£ degli Studi di Torino

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)copy SMILEScopy InChI
Affinity DataKi:  494nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4R0NPubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Eli Lilly and Company Ltd

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)copy SMILEScopy InChI
Affinity DataKi:  789nMAssay Description:Binding affinity of compound was determined against Ionotropic glutamate receptor ionotropic kainate 3 using cell membranes prepared from HEK293 cell...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2765FVBPubMed