Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Glutaminase kidney isoform, mitochondrial' and Ligand = 'BDBM405062'
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM405062(1-[2-fluoro-4-(4-{2-[3- (trifluoromethoxy)phenyl]a...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z76GPUS Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM405062(1-[2-fluoro-4-(4-{2-[3- (trifluoromethoxy)phenyl]a...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2765HQCUS Patent