Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Glycine receptor subunit alpha-1/beta' and Ligand = 'BDBM50232897'
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232897(CHEMBL4068867)copy SMILEScopy InChI
Affinity DataIC50: 116nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232897(CHEMBL4068867)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232897(CHEMBL4068867)copy SMILEScopy InChI
Affinity DataIC50: 355nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed