Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Glycine receptor subunit alpha-1' and Ligand = 'BDBM50232884'
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [3H]strychnine from glycine receptor alpha 1 in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)copy SMILEScopy InChI
Affinity DataIC50: 76nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)copy SMILEScopy InChI
Affinity DataIC50: 77nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)copy SMILEScopy InChI
Affinity DataIC50: 78nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed