Found 4 Enz. Inhib. hit(s) with Target = 'Glycine receptor subunit alpha-1' and Ligand = 'BDBM50232890' TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 189nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataIC50: 105nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
