Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Glycine receptor subunit alpha-1' and Ligand = 'BDBM50510757'
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50510757(CHEMBL4518537)copy SMILEScopy InChI
Affinity DataKi:  91nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571GB7PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50510757(CHEMBL4518537)copy SMILEScopy InChI
Affinity DataIC50: 173nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced whole cell currents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571GB7PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50510757(CHEMBL4518537)copy SMILEScopy InChI
Affinity DataIC50: 708nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571GB7PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50510757(CHEMBL4518537)copy SMILEScopy InChI
Affinity DataIC50: 710nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571GB7PubMed