Found 3 Enz. Inhib. hit(s) with Target = 'Growth hormone secretagogue receptor type 1' and Ligand = 'BDBM50165591' TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier
Curated by ChEMBL
Universit£ de Montpellier
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier
Curated by ChEMBL
Universit£ de Montpellier
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human GHS-R1a transfected in mouse LTK cells after 6 hrs by CRE/luciferase reporter gene assay in presence of ghrelin and roli...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier
Curated by ChEMBL
Universit£ de Montpellier
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human GHS-R1a transfected in CHO cells assessed as inhibition of ghrelin-induced intracellular calcium mobilization measured o...More data for this Ligand-Target Pair
