Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Growth hormone secretagogue receptor type 1' and Ligand = 'BDBM50208678'
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS-Universités Montpellier I et II

Curated by ChEMBL
LigandPNGBDBM50208678((R)-N-(1-(4-(4-methoxybenzyl)-5-(3-phenylpropyl)-4...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251HW6PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS-Universités Montpellier I et II

Curated by ChEMBL
LigandPNGBDBM50208678((R)-N-(1-(4-(4-methoxybenzyl)-5-(3-phenylpropyl)-4...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM586CPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS-Universités Montpellier I et II

Curated by ChEMBL
LigandPNGBDBM50208678((R)-N-(1-(4-(4-methoxybenzyl)-5-(3-phenylpropyl)-4...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Antagonist activity at human GHSR1a receptor expressed in CHO cells assessed as reduction of ghrelin-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM586CPubMed