Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H2 receptor' and Ligand = 'BDBM50568763'
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50568763(CHEMBL4852212)copy SMILES
Affinity DataKi:  100nMAssay Description:Displacement of [3H]UR-DE257 from human histamine H2 receptor expressed in sf9 insect cell membranes co-expressing GSalphaS incubated for 60 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TF0245PubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))TBA
LigandPNGBDBM50568763(CHEMBL4852212)copy SMILES
Affinity DataEC50:  26nMAssay Description:Agonist activity at guinea pig right atrium histamine H2 receptor assessed as increase in heart rate incubated for 30 mins in presence of cimetidineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TF0245PubMed