Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Histamine H2 receptor' and Ligand = 'BDBM50568773'
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50568773(CHEMBL4853772)copy SMILES
Affinity DataKi:  115nMAssay Description:Displacement of [3H]UR-DE257 from human histamine H2 receptor expressed in sf9 insect cell membranes co-expressing GSalphaS incubated for 60 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TF0245PubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50568773(CHEMBL4853772)copy SMILES
Affinity DataEC50:  372nMAssay Description:Agonist activity at human histamine H2 receptor expressed in HEK293T cells co-expressing ELucC by beta arrestin2 recruitment assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TF0245PubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))TBA
LigandPNGBDBM50568773(CHEMBL4853772)copy SMILES
Affinity DataEC50:  89nMAssay Description:Agonist activity at guinea pig right atrium histamine H2 receptor assessed as increase in heart rate incubated for 30 mins in presence of cimetidineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TF0245PubMed