Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM159248'
TargetHistamine H3 receptor(Homo sapiens (Human))
NOVARTIS AG

US Patent
LigandPNGBDBM159248(US9034874, 1.5)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:The potency of compounds of the invention as H3 receptor antagonists can be assessed by measuring the blockade of (R)-alpha-methylhistamine-mediated ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C82819US Patent
TargetHistamine H3 receptor(GUINEA PIG)
Palack£ University

Curated by ChEMBL
LigandPNGBDBM159248(US9034874, 1.5)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Inhibition of Guinea Pig Ileum H3RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41VXGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
Palack£ University

Curated by ChEMBL
LigandPNGBDBM159248(US9034874, 1.5)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Inhibition of Guinea Pig Ileum H3RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41VXGPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
NOVARTIS AG

US Patent
LigandPNGBDBM159248(US9034874, 1.5)copy SMILEScopy InChI
Affinity DataKi:  25nMpH: 7.5Assay Description:The affinity of compounds of the invention to the H3 receptor can be assessed by measuring displacement of binding of the radioligand [3H]-N-alpha -M...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C82819US Patent