Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50139407'
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50139407(4-{2-[2-((2R,6S)-2,6-Dimethyl-piperidin-1-yl)-ethy...)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Binding potency was determined by displacement of [3H]-N-alpha-methyl histamine from cloned human histamine H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20C4V5HPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50139407(4-{2-[2-((2R,6S)-2,6-Dimethyl-piperidin-1-yl)-ethy...)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Binding potency was determined by displacement of [3H]N-alpha-methyl histamine from cloned human histamine H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20C4V5HPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50139407(4-{2-[2-((2R,6S)-2,6-Dimethyl-piperidin-1-yl)-ethy...)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Binding potency was determined by displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20C4V5HPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50139407(4-{2-[2-((2R,6S)-2,6-Dimethyl-piperidin-1-yl)-ethy...)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Binding potency was determined by displacement of [3H]N-alpha-methyl histamine from histamine H3 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20C4V5HPubMed