Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50237879'
TargetHistamine H3 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50237879(2-(1,3-bis(2-(piperidin-1-yl)ethyl)imidazolidin-2-...)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned histamine H3 receptor expressed in monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5FSFPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50237879(2-(1,3-bis(2-(piperidin-1-yl)ethyl)imidazolidin-2-...)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Binding affinity to histamine H3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J9699QPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Kyowa Hakko Kogyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50237879(2-(1,3-bis(2-(piperidin-1-yl)ethyl)imidazolidin-2-...)copy SMILEScopy InChI
Affinity DataKi:  55nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from histamine H3 receptor in rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5FSFPubMed