Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50281388'
TargetHistamine H3 receptor(Homo sapiens (Human))
IQOG, CSIC

Curated by ChEMBL
LigandPNGBDBM50281388(CHEMBL4173258)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human H3R expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN699QPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
IQOG, CSIC

Curated by ChEMBL
LigandPNGBDBM50281388(CHEMBL4173258)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222Z25PubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
IQOG, CSIC

Curated by ChEMBL
LigandPNGBDBM50281388(CHEMBL4173258)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Binding affinity to human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5X88PubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
IQOG, CSIC

Curated by ChEMBL
LigandPNGBDBM50281388(CHEMBL4173258)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human H3R expressed in HEK293 cell membranes incubated for 90 mins by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87F3NPubMed