Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50392759'
TargetHistamine H3 receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50392759(CHEMBL2151157)copy SMILEScopy InChI
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]N-alpha-Methylhistamine from human recombinant H3 receptor expressed in HEK293 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222WCCPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50392759(CHEMBL2151157)copy SMILEScopy InChI
Affinity DataKi:  0.316nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ33RVPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50392759(CHEMBL2151157)copy SMILEScopy InChI
Affinity DataIC50: 2.51nMAssay Description:Inverse agonist activity at human histamine H3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ33RVPubMed