Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase KAT2B [719-832]' and Ligand = 'BDBM311422'
TargetHistone acetyltransferase KAT2B [719-832](Homo sapiens (Human))
GENENTECH, INC; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM311422(US10155764, Example 15A)copy SMILEScopy InChI
Affinity DataIC50: 78nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25M67T9US Patent