TargetHistone deacetylase 1(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Inhibition of human HDAC1More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 0.480nMAssay Description:Inhibition of human recombinant HDAC1 using Fluor de Lys as substrate after 2 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Inhibition of human recombinant HDAC1 using fluorogenic HDAC substrate after 15 mins by fluorimetrc methodMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human HDAC1 expressed in baculovirus infected sf9 cells using p53 residues 379-382 (RHKKAc) as substrate by fluorescence-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
TargetHistone deacetylase 1(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataIC50: 0.110nMAssay Description:Inhibition of full length recombinant human HDAC1 expressed in baculovirus infected Sf9 cells using RHKK-Ac as substrate by fluorescence analysisMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataIC50: 0.110nMAssay Description:Inhibition of recombinant full length C-terminal FLAG His-tagged human HDAC1 expressed in baculovirus infected Sf21 insect cells using RHK-K(Ac)-AMC ...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataIC50: 0.460nMAssay Description:Inhibition of recombinant human full length C-terminal His/FLAG tagged HDAC1 (1 to 482 residues) expressed in baculovirus-infected Sf9 cells using Ac...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataIC50: 0.460nMAssay Description:Inhibition of C-terminal His/Flag-tagged human HDAC1 (1 to 482 residues) expressed in Sf9 cells using Ac-peptide as substrate preincubated for 15 min...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataIC50: 0.617nMAssay Description:Inhibition of recombinant full length human HDAC1 expressed in baculovirus infected Sf9 cells using FAM-RHKK-Ac as substrate incubated for 17 hrs by ...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataIC50: 0.620nMAssay Description:Inhibition of recombinant full length human HDAC1 expressed in SF9 baculovirus using FAM- labelled acetylated peptide as substrate measured by Electr...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
TargetHistone deacetylase 1(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
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