TargetHistone deacetylase 4(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Inhibition of human HDAC4More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 6.70nMAssay Description:Inhibition of human recombinant HDAC4 using fluorogenic HDAC substrate class 2a after 30 mins by fluorimetrc methodMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human HDAC4 expressed in baculovirus infected sf9 cells using (Boc-Lys(trifluoroacetyl)-AMC) as substrate by fluorescence-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
TargetHistone deacetylase 4(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Inhibition of recombinant full length human HDAC4 expressed in SF9 baculovirus using FAM- labelled acetylated peptide as substrate measured by Electr...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
St Jude Children's Research Hospital
Curated by ChEMBL
St Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Inhibition of recombinant full length human HDAC4 expressed in baculovirus infected Sf9 cells using FAM-RHKK-TFAc as substrate incubated for 1.5 hrs ...More data for this Ligand-Target Pair