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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase, H3 lysine-79 specific' and Ligand = 'BDBM50551137'
Target
Histone-lysine N-methyltransferase, H3 lysine-79 specific
(Homo sapiens (Human))
TBA
Ligand
BDBM50551137
(CHEMBL4765125)
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Affinity Data
IC50: 1.00E+3nM
Assay Description:
Inhibition of recombinant human N-terminal GST-tagged DOT1L (1 to 420 residues) expressed in Escherichia coli BL21 (DE3) using histone as substrate i...
More data for this Ligand-Target Pair
Target Info
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MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
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Ligand Info
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MCE
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In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2TB1BJ6
PubMed