Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase EHMT1' and Ligand = 'BDBM50353128'
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Mercachem BV

Curated by ChEMBL
LigandPNGBDBM50353128(CHEMBL1231795)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of N-terminal GST tagged human recombinant EHMT1 (794 to 1294 residues) expressed in baculovirus infected Sf9 insect cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1Q8XPubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Mercachem BV

Curated by ChEMBL
LigandPNGBDBM50353128(CHEMBL1231795)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of EHMT1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC135PPubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Mercachem BV

Curated by ChEMBL
LigandPNGBDBM50353128(CHEMBL1231795)copy SMILEScopy InChI
Affinity DataIC50: 19nMMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Mercachem BV

Curated by ChEMBL
LigandPNGBDBM50353128(CHEMBL1231795)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2280C10PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Mercachem BV

Curated by ChEMBL
LigandPNGBDBM50353128(CHEMBL1231795)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Competitive inhibition of GLP by fluorescence polarization assay in presence of fluorescein-labeled H3 peptideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ62NXPubMed