Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase EHMT1' and Ligand = 'BDBM50446376'
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Mercachem BV

Curated by ChEMBL
LigandPNGBDBM50446376(CHEMBL3109630)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of N-terminal GST tagged human recombinant EHMT1 (794 to 1294 residues) expressed in baculovirus infected Sf9 insect cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1Q8XPubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Mercachem BV

Curated by ChEMBL
LigandPNGBDBM50446376(CHEMBL3109630)copy SMILEScopy InChI
Affinity DataIC50: 38nMMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Mercachem BV

Curated by ChEMBL
LigandPNGBDBM50446376(CHEMBL3109630)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of GLP (unknown origin)-mediated incorporation of methyl group from [3H]-SAM into peptide substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NJ0PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Mercachem BV

Curated by ChEMBL
LigandPNGBDBM50446376(CHEMBL3109630)copy SMILEScopy InChI
Affinity DataIC50: 118nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9H28PubMed