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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase EZH2 [A687V]' and Ligand = 'BDBM190204'
Target
Histone-lysine N-methyltransferase EZH2 [A687V]
(Homo sapiens (Human))
Epizyme, Inc.
US Patent
Ligand
BDBM190204
(EPZ008491 | US9175331, 35)
copy SMILES
Affinity Data
IC50: 2.90nM
Assay Description:
Test compounds were serially diluted 3-fold in DMSO in a 10 point-curve and 1 uL was spotted into a 384-well microplate in duplicate using a Platemat...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2ZW1JQP
US Patent