Found 2 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase SETD2' and Ligand = 'BDBM50582884' 
Affinity DataIC50: 147nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Affinity DataIC50: 449nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
