Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Homeodomain-interacting protein kinase 1' and Ligand = 'BDBM50550127'
TargetHomeodomain-interacting protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50550127(CHEMBL4781866)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human HIPK1 (158 to 555 residues) using myelin ba as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scinti...More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251NSHPubMed
TargetHomeodomain-interacting protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50550127(CHEMBL4781866)copy SMILES
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to human HIPK1 (158 to 555 residues) using myelin ba as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric ...More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251NSHPubMed