Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Homeodomain-interacting protein kinase 3' and Ligand = 'BDBM50537742'
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human His-tagged HIPK3 catalytic domain expressed in baculovirus expression system using serine/threonine-9 peptide as subs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed