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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Inhibitor of nuclear factor kappa-B kinase subunit alpha' and Ligand = 'BDBM27492'
Target
Inhibitor of nuclear factor kappa-B kinase subunit alpha
(Homo sapiens (Human))
GSK
Ligand
BDBM27492
(2-amino-5-phenyl-3-(4-{[2-(pyrrolidin-1-yl)ethyl]s...)
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Affinity Data
IC50: 794nM
Assay Description:
IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2QZ289W
PubMed