Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Insulin-like growth factor 1 receptor' and Ligand = 'BDBM50256468'
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50256468(CHEMBL500003 | N-(2,6-difluorophenyl)-3-(3-(2-(4-(...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of GST-tagged IGF1R (957-1367) (unknown origin) expressed in baculovirus by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6J8MPubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50256468(CHEMBL500003 | N-(2,6-difluorophenyl)-3-(3-(2-(4-(...)copy SMILEScopy InChI
Affinity DataIC50: 174nMAssay Description:Inhibition of human IGF1R autophosphorylation in transfected mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6J8MPubMed